- CARM1 Preferentially Methylates H3R17 over H3R26 through a Random Kinetic Mechanism
Suzanne L. Jacques et al, 2016, Biochemistry CrossRef - Targeting epigenetic regulators for cancer therapy: modulation of bromodomain proteins, methyltransferases, demethylases, and microRNAs
Kathy A. Gelato et al, 2016, Expert Opinion on Therapeutic Targets CrossRef - Identification of a CARM1 Inhibitor with Potent In Vitro and In Vivo Activity in Preclinical Models of Multiple Myeloma
Allison E. Drew et al, 2017, Sci Rep CrossRef - CARM1 Is Essential for Myeloid Leukemogenesis but Dispensable for Normal Hematopoiesis
Sarah M. Greenblatt et al, 2018, Cancer Cell CrossRef - Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 Against Acute Myeloid Leukemia
Zuhao Guo et al, 2019, J. Med. Chem. CrossRef - Differential CARM1 Isoform Expression in Subcellular Compartments and among Malignant and Benign Breast Tumors
David Shlensky et al, 2015, PLoS ONE CrossRef - null
Thomas B. Nicholson et al, 2015 CrossRef - null
Amit K. Behera et al, 2019 CrossRef - Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1
Matthijs J. van Haren et al, 2017, Proc Natl Acad Sci USA CrossRef - AMPK-ERK/CARM1 Signaling Pathways Affect Autophagy of Hepatic Cells in Samples of Liver Cancer Patients
Qiu-Fang Qin et al, 2019, Front. Oncol. CrossRef - Structural and biochemical evaluation of bisubstrate inhibitors of protein arginine N-methyltransferases PRMT1 and CARM1 (PRMT4)
Emma A. Gunnell et al, 2020 CrossRef - null
Matthijs J. van Haren et al, 2019 CrossRef - Protein arginine methylation/demethylation and cancer
Coralie Poulard et al, 2016, Oncotarget CrossRef - CARM1 inhibition reduces histone acetyltransferase activity causing synthetic lethality in CREBBP/EP300-mutated lymphomas
Kylee J. Veazey et al, 2020, Leukemia CrossRef - Epigenetic Aberrations in Multiple Myeloma.
Cinzia Caprio et al, 2020, Cancers (Basel) CrossRef - Arginine Methylation in Brain Tumors: Tumor Biology and Therapeutic Strategies
Jean-Paul Bryant et al, 2021, Cells CrossRef - Protein arginine methyltransferases and hepatocellular carcinoma: A review
Yu Lei et al, 2021, Translational Oncology CrossRef - Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy
Zhuqing Zhang et al, 2021, J. Med. Chem. CrossRef - Ribavirin inhibits the growth and ascites formation of hepatocellular carcinoma through downregulation of type I CARM1 and type II PRMT5
Yizhen Tian et al, 2021, Toxicology and Applied Pharmacology CrossRef - Systematic pan-cancer landscape identifies CARM1 as a potential prognostic and immunological biomarker
Yingqi Qiu et al, 2022, BMC Genom Data CrossRef - Expression of pluripotency-related genes in human glioblastoma
Álvaro Fabrício Lopes Rios et al, 2022 CrossRef - Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction–Reconstruction and Fragment-Growing Approach
Giulia Iannelli et al, 2022, J. Med. Chem. CrossRef - Protein Arginine Methyltransferases (PRMTs): Orchestrators of Cancer Pathogenesis, Immunotherapy Dynamics, and Drug Resistance
Yihang Gao et al, 2024, Biochemical Pharmacology CrossRef - Development of (2-(Benzyloxy)phenyl)methanamine Derivatives as Potent and Selective Inhibitors of CARM1 for the Treatment of Melanoma
Zhihao Liu et al, 2024, J. Med. Chem. CrossRef - Tyrosine phosphorylation of CARM1 promotes its enzymatic activity and alters its target specificity
Hidehiro Itonaga et al, 2024, Nat Commun CrossRef